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Active

Caffeine

Caffeine is a active, antioxidant, skin conditioning used in cosmetic and personal-care formulation. Typical use level is 0.5%–3%. It is water-soluble. Stable in the pH 4–7 range.

At a glance

CAS number
58-08-2
INCI name
Caffeine
Function
active, antioxidant, skin conditioning
Typical use level
0.5%–3%
Solubility
water
Stable pH
4–7

CAS number and synonyms are sourced from PubChem. Function, usage levels, pH and compatibility are AI-assisted formulation guidance — verify against your supplier's technical data sheet and applicable regulations before use.

Also known as

caffeine Guaranine 1,3,7-Trimethylxanthine Methyltheobromine Theine Thein Cafeina Caffein Cafipel Koffein Mateina Alert-pep

Compatibility

Works well with:
Niacinamide Hyaluronic Acid Glycerin Panthenol Allantoin Green Tea Extract Retinol Peptides Vitamin E

Use caution with:
Tannic Acid High-concentration Tannins Strong Oxidizing Agents

Caffeine can form insoluble complexes with tannins and polyphenols at higher concentrations, potentially causing precipitation or reduced efficacy. It is generally stable and compatible with most common cosmetic actives across a moderate pH range. Strong oxidizing agents may degrade the xanthine structure over time.

Formulation notes

No specific regulatory maximum in EU cosmetics; typical use is 0.5–3% in eye creams, serums, and slimming products. Solubility in water is approximately 20 mg/mL at room temperature (2%), so formulations above this level may require warming or a co-solvent. No known sensitization concerns at typical use levels.

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